Save up -80% on Cyclobenzaprine
Note: this is a drug discount program, not an insurance plan.
2018 Price of Cyclobenzaprine
Cyclobenzaprine 5 mg tablet
* price without discount in nearest pharmacy. Price may vary.
We offer free Cyclobenzaprine coupons and discounts that may help you save up to 80% off the retail price in your local pharmacy. Just print your coupon! It’s ready to use and never expire. Present your discount card in most local pharmacies to get a discount on Cyclobenzaprine every time. What are you waiting for? Claim your prescription drug card now!
Cyclobenzaprine volume of distribution
Discount Cards 16,000+
Clients Benefit 29%
Total savings $4,735,080
What is Cyclobenzaprine
Cyclobenzaprine is a skeletal muscle relaxant and a central nervous system (CNS) depressant. Cyclobenzaprine acts on the locus coeruleus where it results in increased norepinephrine release, potentially through the gamma fibers which innervate and inhibit the alpha motor neurons in the ventral horn of the spinal cord. It is structurally similar to Amitriptyline, differing by only one double bond.
Cyclobenzaprine mechanism of action
Like other tricyclic antidepressants, cyclobenzaprine exhibits anticholinergic activity, potentiation of norepinephrine, and antagonism of reserpine. Cyclobenzaprine does not directly act on the neuromuscular junction or the muscle but relieves muscle spasms through a central action, possibly at the brain stem level. Cyclobenzaprine binds to the serotonin receptor and is considered a 5-HT2 receptor antagonist that reduces muscle tone by decreasing the activity of descending serotonergic neurons.
Dosage forms of Cyclobenzaprine
|Capsule, extended release||oral||15 mg/1|
|Capsule, extended release||oral||30 mg/1|
Alti-cyclobenzaprine – Tab 10mg
Altimed Pharma Inc.
Humans and other mammals
Toxicity of Cyclobenzaprine
Oral mouse and rat LD sub 50 /sub are 338 mg/kg and 425 mg/kg respectively. Signs of overdose include agitation, coma, confusion, congestive heart failure, convulsions, dilated pupils, disturbed concentration, drowsiness, hallucinations, high or low temperature, increased heartbeats, irregular heart rhythms, muscle stiffness, overactive reflexes, severe low blood pressure, stupor, and vomiting.
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