Save up -80% on Eletriptan

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RX BIN: 015558RX PCN: HTGroup ID: DDN6600Card Holder ID: DDN6600
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2019 Price of Relpax

$57.516 tablets/40 mg
Price with discount in nearest pharmacy. Price may vary.

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We offer free Relpax coupons and discounts that may help you save up to 80% off the retail price in your local pharmacy. Just print your coupon! It’s ready to use and never expire. Present your manufacturer copay card in most local pharmacies to get a discount on Eletriptan every time. What are you waiting for? Claim your prescription drug card now!

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Eletriptan volume of distribution

The volume of distribution of eletriptan following IV administration is 138L. Plasma protein binding is moderate and approximately 85%.

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2018 Statistics

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Discount Cards 16,000+

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Clients Benefit 29%

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Total savings $4,735,080

What is Eletriptan

Eletriptan is a second generation triptan drug developed by Pfizer Inc for the treatment of migraine headaches. (Wikipedia)

Eletriptan mechanism of action

Eletriptan binds with high affinity to 5-HT1B, 5-HT1D and 5-HT1F receptors, has modest affinity for 5-HT1A, 5-HT1E, 5-HT2B and 5-HT7 receptors, and little or no affinity for 5-HT2A, 5-HT2C, 5-HT3, 5-HT4, 5-HT5A and 5-HT6 receptors. Eletriptan has no significant affinity or pharmacological activity at adrenergic alpha1, alpha2, or beta; dopaminergic D1 or D2; muscarinic; or opioid receptors. Two theories have been proposed to explain the efficacy of 5-HT receptor agonists in migraine. One theory suggests that activation of 5-HT1 receptors located on intracranial blood vessels, including those on the arteriovenous anastomoses, leads to vasoconstriction, which is correlated with the relief of migraine headache. The other hypothesis suggests that activation of 5-HT1 receptors on sensory nerve endings in the trigeminal system results in the inhibition of pro-inflammatory neuropeptide release.

Dosage forms of Eletriptan

DrugDosageQuantityPrice
Relpax20mg12 Tablet$155.00
Relpax40mg6 Tablet$68.00
Relpax40mg24 Tablet$240.00
Eletriptan20mg6 Tablet$56.75
Eletriptan20mg6 Tablet$56.75

Prescription Generics

true

International Brands

Apo-eletriptan

Synonyms

Eletriptanum

Manufacturers

Apotex Inc

CAS number

143322-58-1

UNII

22QOO9B8KI

State

solid

Affected organisms

Humans and other mammals

Indication of Eletriptan

For the acute treatment of migraine with or without aura in adults.

Toxicity of Eletriptan

Based on the pharmacology of the 5-HT1B/1D agonists, hypertension or other more serious cardiovascular symptoms could occur on overdose.

RX24 Drugs Disclaimer: consult your healthcare provider before buying a Eletriptan on prescription or using an RX manufacturer savings coupon. Content on this page is provided for informational purposes only. Any use of this information is at your own risk.

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What is Relpax?

Relpax is referred to selective serotonin receptor agonists of types 5-HT1B and 5-HT1D-receptors located in cerebral vessels, on the neurons of the nucleus and on the endings of the nervus trigeminus, respectively. In addition to impaired excretion of algogenic substances from nerve endings, Relpax causes vasoconstriction of the cranial vessels. The drug helps to increase the threshold sensitivity of the trigeminal nerve by blocking its spinal nuclei. Clinically, the effect of Relpax is manifested by a decrease in the pulsation of the cerebral vessels, the elimination of pain syndrome.

Relpax, unlike other representatives of triptans, lacks the ability to interact with muscarinic, dopamine, alpha, beta-adrenergic and opioid receptors. After oral administration of Relpax tablets, the active ingredient is immediately absorbed through the intestinal wall, and then binds to plasma proteins by 85%. Tmax after oral pills averaged 1.5 hours. The metabolism of eletriptan, the active ingredient of Relpax, is carried out in the liver by CYP3A4 cytochrome P450. Excretion of metabolites is carried out by the kidneys and gastrointestinal tract.

Relpax should be taken as early as possible, however, the drug is effective at a later stage of a migraine attack. The recommended starting dose is 40 mg. If migraine headache resumes within 24 hours, then Relpax® can be prescribed again in the same dose. If a second dose is needed, it should be taken no earlier than 2 hours after the first dose. The daily dose should not exceed 160 mg.