Save up -80% on Eletriptan
Note: this is a drug discount program, not an insurance plan.
2018 Price of Eletriptan
Relpax 20 mg tablet
* price without discount in nearest pharmacy. Price may vary.
We offer free Eletriptan coupons and discounts that may help you save up to 80% off the retail price in your local pharmacy. Just print your coupon! It’s ready to use and never expire. Present your discount card in most local pharmacies to get a discount on Eletriptan every time. What are you waiting for? Claim your prescription drug card now!
Eletriptan volume of distribution
* 138 L
Discount Cards 16,000+
Clients Benefit 29%
Total savings $4,735,080
What is Eletriptan
Eletriptan is a second generation triptan drug developed by Pfizer Inc for the treatment of migraine headaches. (Wikipedia)
Eletriptan mechanism of action
Eletriptan binds with high affinity to 5-HT1B, 5-HT1D and 5-HT1F receptors, has modest affinity for 5-HT1A, 5-HT1E, 5-HT2B and 5-HT7 receptors, and little or no affinity for 5-HT2A, 5-HT2C, 5-HT3, 5-HT4, 5-HT5A and 5-HT6 receptors. Eletriptan has no significant affinity or pharmacological activity at adrenergic alpha1, alpha2, or beta; dopaminergic D1 or D2; muscarinic; or opioid receptors. Two theories have been proposed to explain the efficacy of 5-HT receptor agonists in migraine. One theory suggests that activation of 5-HT1 receptors located on intracranial blood vessels, including those on the arteriovenous anastomoses, leads to vasoconstriction, which is correlated with the relief of migraine headache. The other hypothesis suggests that activation of 5-HT1 receptors on sensory nerve endings in the trigeminal system results in the inhibition of pro-inflammatory neuropeptide release.
Dosage forms of Eletriptan
|Tablet, film coated||oral||20 mg/1|
Humans and other mammals
Indication of Eletriptan
For the acute treatment of migraine with or without aura in adults.
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