Save up -80% on Fulvestrant
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Price of Fulvestrant
Faslodex 125 mg/2.5 ml syringe
* price without discount in nearest pharmacy. Price may vary.
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Fulvestrant volume of distribution
* 3 to 5 L/kg
What is Fulvestrant
Fulvestrant is a drug treatment of hormone receptor-positive metastatic breast cancer in post-menopausal women with disease progression following anti-estrogen therapy. It is an estrogen receptor antagonist with no agonist effects, which works both by down-regulating and by degrading the estrogen receptor.
Fulvestrant mechanism of action
Fulvestrant competitively and reversibly binds to estrogen receptors present in cancer cells and achieves its anti-estrogen effects through two separate mechanisms. First, fulvestrant binds to the receptors and downregulates them so that estrogen is no longer able to bind to these receptors. Second, fulvestrant degrades the estrogen receptors to which it is bound. Both of these mechanisms inhibit the growth of tamoxifen-resistant as well as estrogen-sensitive human breast cancer cell lines.
Dosage forms of Fulvestrant
|Solution for injection||Intramuscular use||250 mg/5ml|
Astra Zeneca Pharmaceuticals Lp
Humans and other mammals
Indication of Fulvestrant
For the treatment of hormone receptor positive metastatic breast cancer in postmenopausal women with disease progression following anti-estrogen therapy.
Toxicity of Fulvestrant
There is no clinical experience with overdosage in humans.
Disclaimer: before buying a Fulvestrant on prescription, consult your health care provider. Content on this page is provided for informational purposes only. Any use of this information is at your own risk.