Save up -80% on Naltrexone

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RX BIN: 015558
RX PCN: HT
Group ID: DDN6600
Card Holder ID: DDN6600

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2018 Price of Naltrexone

Depade 50 mg tablet

$4.28

tablet

* price without discount in nearest pharmacy. Price may vary.

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Naltrexone volume of distribution

* 1350 L (intravenous administration)

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What is Naltrexone

Derivative of noroxymorphone that is the N-cyclopropylmethyl congener of naloxone. It is a narcotic antagonist that is effective orally, longer lasting and more potent than naloxone, and has been proposed for the treatment of heroin addiction. The FDA has approved naltrexone for the treatment of alcohol dependence.

Naltrexone mechanism of action

Naltrexone is a pure opiate antagonist and has little or no agonist activity. The mechanism of action of naltrexone in alcoholism is not understood; however, involvement of the endogenous opioid system is suggested by preclinical data. Naltrexone is thought to act as a competitive antagonist at mc, , and receptors in the CNS, with the highest affintiy for the receptor. Naltrexone competitively binds to such receptors and may block the effects of endogenous opioids. This leads to the antagonization of most of the subjective and objective effects of opiates, including respiratory depression, miosis, euphoria, and drug craving. The major metabolite of naltrexone, 6–naltrexol, is also an opiate antagonist and may contribute to the antagonistic activity of the drug.

Dosage forms of Naltrexone

DrugDosageQuantityPrice
Revia50mg50 Tablet$379.00
Naltrexone50mg30 Tablet$79.00
Naltrexone50mg90 Tablet$218.00
Prescription Generics

true

International Brands

Apo-naltrexone

Synonyms

17-(Cyclopropylmethyl)-4,5-epoxy-3,14-dihydroxymorphinan-6-one 17-(Cyclopropylmethyl)-4,5alpha-epoxy-3,14-dihydroxymorphinan-6-one

Manufacturers

Apotex Inc

CAS number

16590-41-3

UNII

5S6W795CQM

State

solid

Affected organisms

Humans and other mammals

Indication of Naltrexone

Used as an adjunct to a medically supervised behaviour modification program in the maintenance of opiate cessation in individuals who were formerly physically dependent on opiates and who have successfully undergone detoxification. Also used for the management of alcohol dependence in conjunction with a behavioural modification program.

Toxicity of Naltrexone

In the mouse, rat and guinea pig, the oral LD sub50 /subs were 1,100-1,550 mg/kg; 1,450 mg/kg; and 1,490 mg/kg; respectively. High doses of naltrexone (generally ge;1,000 mg/kg) produce salivation, depression/reduced activity, tremors, and convulsions.

RX24 Drugs Disclaimer: before buying a Naltrexone on prescription, consult your healthcare provider. Content on this page is provided for informational purposes only. Any use of this information is at your own risk.

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