Save up -80% on Sulfinpyrazone
Note: this is a drug discount program, not an insurance plan.
Pharmacists and Patients support.
2018 Price of Sulfinpyrazone
Apo-Sulfinpyrazone 200 mg Tablet
tablet
* price without discount in nearest pharmacy. Price may vary.
Claim your free Sulfinpyrazone discount card
We offer free Sulfinpyrazone coupons and discounts that may help you save up to 80% off the retail price in your local pharmacy. Just print your coupon! It’s ready to use and never expire. Present your discount card in most local pharmacies to get a discount on Sulfinpyrazone every time. What are you waiting for? Claim your prescription drug card now!
Sulfinpyrazone volume of distribution
About RX24Drugs
Discount Cards 16,000+
Clients Benefit 29%
Total savings $4,735,080
Sulfinpyrazone mechanism of action
Sulfinpyrazone is an oral uricosuric agent (pyrazolone derivative) used to treat chronic or intermittent gouty arthritis. Sulfinpyrazone competitively inhibits the reabsorption of uric acid at the proximal convoluted tubule, thereby facilitating urinary excretion of uric acid and decreasing plasma urate concentrations. This is likely done through inhibition of the urate anion transporter (hURAT1) as well as the human organic anion transporter 4 (hOAT4). Sulfinpyrazone is not intended for the treatment of acute attacks because it lacks therapeutically useful analgesic and anti-inflammatory effects. Sulfinpyrazone and its sulfide metabolite possess COX inhibitory effects. Sulfinpyrazone has also been shown to be a UDP-glucuronsyltransferase inhibitor and a very potent CYP2C9 inhibitor. Sulfinpyrazone is also known to be a cystic fibrosis transmembrane conductance regulator (CFTR) inhibitor as well as an inhibitor of several multridrug resistance proteins (MRPs).
Dosage forms of Sulfinpyrazone
| Form | Route | Strength |
|---|---|---|
| Tablet | oral | 100 mg |
| Tablet | oral | 200 mg |
Prescription Generics
false
International Brands
Antazone Tab 100mg
Synonyms
1,2-Diphenyl-3,5-dioxo-4-(2-phenylsulfinylethyl)pyrazolidine 1,2-Diphenyl-4-(2′-phenylsulfinethyl)-3,5-pyrazolidinedione
Manufacturers
Icn Canada Ltd.
CAS number
57-96-5
UNII
V6OFU47K3W
State
solid
Affected organisms
Humans and other mammals
Indication of Sulfinpyrazone
For the treatment of gout and gouty arthritis.
RX24 Drugs Disclaimer: before buying a Sulfinpyrazone on prescription, consult your healthcare provider. Content on this page is provided for informational purposes only. Any use of this information is at your own risk.
